SCHEMBL6939399

SCHEMBL6939399

C[C@](C(=O)NN)(c1cccc(C2CCC2)c1[C@H](C/C=C/c1ccccc1)C(=O)NO)S(C)(=O)=O

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.35
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
CTSC P53634 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6943822 0.98 ADAM17 (0.35) ADAM17MMP1MMP9MMP13CTSC
SCHEMBL6943842 0.87 P2RX3 (0.32)
SCHEMBL6942474 0.86 P2RX3 (0.33)
SCHEMBL6939584 0.74 ADAM17 (0.36) ADAM17MMP1MMP9MMP13CTSC
SCHEMBL7937181 0.71 ADAM17 (0.35) ADAM17MMP1MMP9MMP13CTSC
SCHEMBL6939934 0.69 ADAM17 (0.36) ADAM17MMP1MMP9MMP13CTSC
SCHEMBL6940940 0.66 ADAM17 (0.35) ADAM17MMP1MMP9MMP13CTSC
SCHEMBL6943958 0.65 ADAM17 (0.34) ADAM17CTSC
SCHEMBL6944520 0.63 HDAC3 (0.36) ADAM17CTSC
SCHEMBL6942160 0.63 ADAM17 (0.37) ADAM17MMP1MMP9MMP13CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed
EP-0993442-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-04-19 EP disclosed
WO-1999001428-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-01-14 WO disclosed