SCHEMBL6943822

SCHEMBL6943822

C[C@](C(=O)NN)(c1cccc(C2CCCC2)c1[C@H](C/C=C/c1ccccc1)C(=O)NO)S(C)(=O)=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.35
CTSC P53634 1/20 0.33
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
USP2 O75604 1/20 0.32
CYP1A2 P05177 1/20 0.32
HTR1A P08908 1/20 0.32
ADRA2A P08913 1/20 0.32
CYP2D6 P10635 1/20 0.32
CHRM1 P11229 1/20 0.32
CYP2C9 P11712 1/20 0.32
DRD1 P21728 1/20 0.32
TBXA2R P21731 1/20 0.32
PTGS1 P23219 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
ADRA1A P35348 1/20 0.32
OPRM1 P35372 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939399 0.98 ADAM17 (0.35) ADAM17CTSCMMP1MMP9MMP13
SCHEMBL6942474 0.88 P2RX3 (0.33)
SCHEMBL6943842 0.87 P2RX3 (0.32)
SCHEMBL6939584 0.74 ADAM17 (0.36) ADAM17CTSCMMP1MMP9MMP13
SCHEMBL7937181 0.72 ADAM17 (0.35) ADAM17CTSCMMP1MMP9MMP13
SCHEMBL6939934 0.69 ADAM17 (0.36) ADAM17CTSCMMP1MMP9MMP13
SCHEMBL6940940 0.66 ADAM17 (0.35) ADAM17CTSCMMP1MMP9MMP13
SCHEMBL6944520 0.63 HDAC3 (0.36) ADAM17CTSC
SCHEMBL6942160 0.63 ADAM17 (0.37) ADAM17CTSCMMP1MMP9MMP13
SCHEMBL6943958 0.63 ADAM17 (0.34) ADAM17CTSCMASP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed
EP-0993442-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-04-19 EP disclosed
WO-1999001428-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-01-14 WO disclosed