SCHEMBL7937181

SCHEMBL7937181

CS(=O)(=O)c1ccccc1[C@](CC1CCCC1)(C(=O)NN)[C@H](C/C=C/c1ccccc1)C(=O)NO

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 3/20 0.35
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
OPRK1 P41145 1/20 0.34
CTSC P53634 1/20 0.33
MMP1 P03956 2/20 0.33
MMP9 P14780 2/20 0.33
MMP13 P45452 2/20 0.33
MASP2 O00187 1/20 0.33
CHRM3 P20309 1/20 0.31
GCK P35557 1/20 0.30
MMP2 P08253 2/20 0.30
MMP3 P08254 1/20 0.30
BMP1 P13497 1/20 0.30
GRIK1 P39086 1/20 0.30
GRIK2 Q13002 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7937124 0.88 P2RX3 (0.32) ALDH1A1GAAOPRK1
SCHEMBL7937182 0.78 ADAM17 (0.36) ADAM17ALDH1A1GAAOPRK1CTSC
SCHEMBL6977404 0.75 MASP2 (0.36) ADAM17ALDH1A1GAAOPRK1CTSC
SCHEMBL6943822 0.72 ADAM17 (0.35) ADAM17ALDH1A1GAACTSCMMP1
SCHEMBL6983563 0.71 ALDH1A1 (0.33) ADAM17ALDH1A1GAACTSCMMP1
SCHEMBL6939399 0.71 ADAM17 (0.35) ADAM17CTSCMMP1MMP9MMP13
SCHEMBL7937125 0.70 ALDH1A1 (0.31) ALDH1A1GAACTSC
SCHEMBL6986114 0.69 ALDH1A1 (0.31) ADAM17ALDH1A1GAAMMP1MMP9
SCHEMBL6942160 0.67 ADAM17 (0.37) ADAM17CTSCMMP1MMP9MMP13
SCHEMBL6982221 0.67 REN (0.34) ALDH1A1GAACTSCMASP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed