SCHEMBL6940065

SCHEMBL6940065

O=C(O)C(=Cc1ccc(OCc2c(Cl)cccc2Cl)cc1)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.57
ITGA4 P13612 3/20 0.57
SMN1; SMN2 Q16637 2/20 0.49
NR1H4 Q96RI1 1/20 0.47
TP53 P04637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
ALDH1A1 P00352 1/20 0.44
NR4A2 P43354 1/20 0.43
HPGD P15428 2/20 0.42
MAPT P10636 2/20 0.42
MRGPRX4 Q96LA9 1/20 0.41
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
GAA P10253 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7215453 0.88 NR1H4 (0.63) ITGB1ITGA4SMN1; SMN2NR1H4NPSR1
SCHEMBL7215467 0.83 NR1H4 (0.67) ITGB1ITGA4SMN1; SMN2NR1H4NPSR1
SCHEMBL7046284 0.80 SMN1; SMN2 (0.56) ITGB1ITGA4SMN1; SMN2TP53NPSR1
SCHEMBL7046280 0.80 SMN1; SMN2 (0.56) ITGB1ITGA4SMN1; SMN2TP53NPSR1
SCHEMBL6955487 0.79 NR1H4 (0.70) NR1H4TP53NR4A2MAPTKDM4E
SCHEMBL6602394 0.79 SMN1; SMN2 (0.57) ITGB1ITGA4SMN1; SMN2NPSR1KMT2A
SCHEMBL3499309 0.75 NR1H4 (0.58) ITGB1ITGA4SMN1; SMN2NR1H4NR4A2
SCHEMBL7050289 0.74 ITGA4 (0.45) ITGB1ITGA4SMN1; SMN2NR1H4NPSR1
SCHEMBL7017204 0.74 TP53 (0.47) NR1H4TP53
SCHEMBL7483584 0.74 SMN1; SMN2 (0.69) SMN1; SMN2NR1H4KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1206463-A4 FATTY ACID SYNTHASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-01-29 EP disclosed
EP-1206465-A4 FATTY ACID SYNTHASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-01-02 EP disclosed
EP-1206463-A1 FATTY ACID SYNTHASE INHIBITORS SmithKline Beecham Corporation (US) 2002-05-22 EP disclosed
EP-1206465-A1 FATTY ACID SYNTHASE INHIBITORS SmithKline Beecham Corporation (US) 2002-05-22 EP disclosed
WO-2001014364-A1 FATTY ACID SYNTHASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-03-01 WO disclosed
WO-2001014362-A1 FATTY ACID SYNTHASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-03-01 WO disclosed