SCHEMBL6940928

SCHEMBL6940928

CC(C)C[C@](C(=O)NN)([C@H](C(=O)NO)C(/C=C/c1ccccc1)C1CCCCCC1)S(C)(=O)=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
ADAM17 P78536 2/20 0.34
HSP90AA1 P07900 2/20 0.33
HDAC3 O15379 2/20 0.33
HDAC4 P56524 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC7 Q8WUI4 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC10 Q969S8 2/20 0.33
HDAC11 Q96DB2 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
HDAC9 Q9UKV0 2/20 0.33
HDAC5 Q9UQL6 2/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 1/20 0.33
MMP1 P03956 1/20 0.33
MMP3 P08254 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6941959 0.77 P2RX3 (0.34) ALDH1A1GAACTSKLNPEP
SCHEMBL7937957 0.73 P2RX3 (0.33)
SCHEMBL6940930 0.73 ADAM17 (0.40) ALDH1A1GAAADAM17HSP90AA1MAPK1
SCHEMBL7928806 0.70 P2RX3 (0.34) ALDH1A1GAAADAM17LNPEP
SCHEMBL6946037 0.70 ADAM17 (0.41) ALDH1A1GAAADAM17MMP1MMP3
SCHEMBL6942733 0.69 ADAM17 (0.36) GAAADAM17HDAC3HDAC4HDAC1
SCHEMBL6940010 0.69 ADAM17 (0.42) ALDH1A1GAAADAM17POLBMMP1
SCHEMBL6947364 0.69 ADAM17 (0.42) ALDH1A1GAAADAM17POLBMMP1
SCHEMBL6939483 0.68 ADAM17 (0.41) ALDH1A1GAAADAM17MMP1MMP3
SCHEMBL6939940 0.68 ADAM17 (0.42) ALDH1A1GAAADAM17MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed