SCHEMBL6942733

SCHEMBL6942733

CC(C)C[C@](CC(C)(C)C)(C(=O)NN)[C@@H](C(=O)NO)C(/C=C/c1ccccc1)S(C)(=O)=O

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 2/20 0.36
HTT P42858 1/20 0.31
CNR2 P34972 1/20 0.31
MMP1 P03956 3/20 0.31
MMP13 P45452 3/20 0.31
MMP9 P14780 1/20 0.31
HDAC3 O15379 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC7 Q8WUI4 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC10 Q969S8 1/20 0.30
HDAC11 Q96DB2 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
HDAC9 Q9UKV0 1/20 0.30
HDAC5 Q9UQL6 1/20 0.30
MMP2 P08253 2/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6942860 0.71 ADAM17 (0.46) ADAM17HTTMMP1MMP9HDAC3
SCHEMBL6942735 0.70 ADAM17 (0.42) ADAM17HTTMMP1MMP13MMP9
SCHEMBL7931077 0.69 ADAM17 (0.34) ADAM17GAA
SCHEMBL6940928 0.69 ALDH1A1 (0.35) ADAM17MMP1MMP13MMP9HDAC3
SCHEMBL4481740 0.66 ADAM17 (0.46) ADAM17MMP1MMP13MMP9MMP2
SCHEMBL6942610 0.66 ADAM17 (0.46) ADAM17MMP1MMP13MMP9MMP2
SCHEMBL6945777 0.65 ADAM17 (0.47) ADAM17MMP1MMP13MMP9MMP2
SCHEMBL6982009 0.65 ADAM17 (0.43) ADAM17MMP1MMP13MMP9MMP2
SCHEMBL7813083 0.65 ADAM17 (0.43) ADAM17MMP1MMP13MMP9MMP2
SCHEMBL7782662 0.65 ADAM17 (0.37) ADAM17HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed
EP-0993442-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-04-19 EP disclosed
WO-1999001428-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-01-14 WO disclosed