SCHEMBL6940930

SCHEMBL6940930

CC(C)C[C@](C(=O)NNC1CCCCCC1)([C@@H](CC=Cc1ccccc1)C(=O)NO)S(C)(=O)=O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.40
HSP90AA1 P07900 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPK1 P28482 1/20 0.36
POLB P06746 2/20 0.36
GAA P10253 2/20 0.35
ALDH1A1 P00352 1/20 0.35
RAB9A P51151 1/20 0.34
KDM4E B2RXH2 2/20 0.34
CTSC P53634 1/20 0.33
LMNA P02545 3/20 0.32
CHRM3 P20309 1/20 0.32
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7928806 0.76 P2RX3 (0.34) ADAM17GAAALDH1A1CTSC
SCHEMBL7937958 0.74 P2RX3 (0.31) ADAM17
SCHEMBL7940268 0.73 P2RX3 (0.30)
SCHEMBL6940928 0.73 ALDH1A1 (0.35) ADAM17HSP90AA1SMN1; SMN2MAPK1POLB
SCHEMBL8107435 0.72 KMT2A (0.31) ADAM17
SCHEMBL8111767 0.71 GAA (0.33) SMN1; SMN2GAA
SCHEMBL7937824 0.71 SMN1; SMN2 (0.33) SMN1; SMN2
SCHEMBL6942735 0.70 ADAM17 (0.42) ADAM17SMN1; SMN2GAACTSCMMP1
SCHEMBL7937182 0.70 ADAM17 (0.36) ADAM17GAAALDH1A1CTSCCHRM3
SCHEMBL7937724 0.70 P2RX7 (0.36) ADAM17SMN1; SMN2MAPK1POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed