SCHEMBL6943182

SCHEMBL6943182

CCC[C@@](C(C)=O)(C(=O)NN)c1ccc(C)cc1[C@H](C/C=C/c1ccccc1)C(=O)NO

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSC P53634 1/20 0.34
MAPT P10636 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
LMNA P02545 2/20 0.33
HTT P42858 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
TP53 P04637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
PIN1 Q13526 1/20 0.32
GRIK1 P39086 3/20 0.31
GRIK2 Q13002 3/20 0.31
NFE2L2 Q16236 1/20 0.31
ADAM17 P78536 1/20 0.31
HTR2A P28223 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6943055 0.91 PIN1 (0.34) CTSCMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL6985696 0.91 CTSC (0.35) CTSCMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL6943697 0.89 MASP2 (0.34) CTSCMEN1KMT2A
SCHEMBL6987488 0.84 ADAM17 (0.31) CTSCGRIK1GRIK2ADAM17
SCHEMBL6986164 0.84 ADAM17 (0.31) CTSCGRIK1GRIK2ADAM17
SCHEMBL6940940 0.84 ADAM17 (0.35) CTSCMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL6940166 0.84 TGFBR1 (0.34)
SCHEMBL6945559 0.84 PIN1 (0.37) CTSCMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL6942465 0.83 PIN1 (0.32) CTSCMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL6941574 0.82 ADAM17 (0.38) ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed