SCHEMBL6943874

SCHEMBL6943874

Cc1ccc2[nH]cc(CCN(C)C)c2c1.c1cn2n1C2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 10/20 0.58
HTR2C P28335 8/20 0.58
HTR2A P28223 6/20 0.58
SLC6A4 P31645 2/20 0.58
MPO P05164 1/20 0.58
HTR1D P28221 12/20 0.56
HTR1B P28222 9/20 0.56
HTR2B P41595 4/20 0.55
HTR1E P28566 3/20 0.55
HTR7 P34969 3/20 0.55
HTR5A P47898 3/20 0.55
HTR6 P50406 3/20 0.55
HTR3E A5X5Y0 2/20 0.55
HTR3B O95264 2/20 0.55
HTR1F P30939 2/20 0.55
HTR3A P46098 2/20 0.55
HTR4 Q13639 2/20 0.55
HTR3D Q70Z44 2/20 0.55
HTR3C Q8WXA8 2/20 0.55
CYP1A2 P05177 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29633081 0.89 HTR1A (0.70) HTR1AHTR2CHTR2ASLC6A4MPO
SCHEMBL4055413 0.89 HTR1A (0.70) HTR1AHTR2CHTR2ASLC6A4MPO
SCHEMBL7076438 0.88 HTR1D (0.60) HTR1AHTR2CHTR2ASLC6A4MPO
SCHEMBL6945756 0.87 HTR1D (0.50) HTR1AHTR2CHTR2ASLC6A4MPO
SCHEMBL7480335 0.84 HTR1D (0.57) HTR1AHTR2CHTR2ASLC6A4HTR1D
SCHEMBL27374778 0.83 MPO (0.61) HTR1AHTR2CHTR2ASLC6A4MPO
SCHEMBL7478879 0.82 HTR1D (0.55) HTR1AHTR2CHTR2ASLC6A4MPO
SCHEMBL6942952 0.80 HTR1A (0.56) HTR1AHTR2CHTR2ASLC6A4MPO
SCHEMBL7324823 0.79 HTR1D (0.68) HTR1AHTR2CHTR2ASLC6A4MPO
SCHEMBL15701982 0.78 HTR2A (0.70) HTR1AHTR2CHTR2ASLC6A4MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0925302-B1 PALLADIUM CATALYZED INDOLIZATION MERCK & CO INC (US) 2002-11-20 EP claimed
US-5567824-A CATALYZING THE CYCLIZATION IN PRESENCE OF A SOLVENT AND A PROTON ACCEPTOR MERCK & CO., INC. (US) 1996-10-22 US claimed
EP-0763032-B1 PALLADIUM CATALYZED RING CLOSURE OF TRIAZOLYL TRYPTAMINE MERCK & CO INC (US) 2003-10-15 EP disclosed
EP-0925302-B1 PALLADIUM CATALYZED INDOLIZATION MERCK & CO INC (US) 2002-11-20 EP disclosed
US-5567824-A CATALYZING THE CYCLIZATION IN PRESENCE OF A SOLVENT AND A PROTON ACCEPTOR MERCK & CO., INC. (US) 1996-10-22 US disclosed