SCHEMBL6946767

SCHEMBL6946767

Nc1ncc2ncn(CCCCc3ccccc3)c2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.50
HDAC6 Q9UBN7 2/20 0.46
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
ADRA1A P35348 1/20 0.45
HSD17B10 Q99714 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
HTT P42858 1/20 0.43
TMIGD3 P0DMS9 2/20 0.42
ADORA1 P30542 2/20 0.42
CYP2D6 P10635 1/20 0.42
TSHR P16473 1/20 0.41
TLR8 Q9NR97 1/20 0.40
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
ADORA2B P29275 1/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6948072 0.96 ADORA2A (0.54) ADORA2AHDAC6KDM4EALDH1A1HPGD
SCHEMBL6950880 0.91 HTT (0.54) ADORA2AHDAC6KDM4EALDH1A1HPGD
SCHEMBL28299548 0.82 HDAC6 (0.63) ADORA2AHDAC6KDM4EALDH1A1HPGD
SCHEMBL26605342 0.78 ALDH1A1 (0.51) ADORA2AHDAC6KDM4EALDH1A1HPGD
SCHEMBL15879501 0.78 ALDH1A1 (0.51) ADORA2AHDAC6KDM4EALDH1A1HPGD
SCHEMBL6948973 0.77 L3MBTL1 (0.56) HDAC6KDM4EALDH1A1HPGDADRA1A
SCHEMBL14010824 0.74 KDM4E (0.55) ADORA2AHDAC6KDM4EALDH1A1HPGD
SCHEMBL3151968 0.74 KDM4E (0.55) ADORA2AHDAC6KDM4EALDH1A1HPGD
SCHEMBL3157542 0.74 HSD17B10 (0.52) ADORA2AHDAC6KDM4EALDH1A1HPGD
SCHEMBL20509322 0.74 HPRT1 (0.55) HDAC6KDM4EALDH1A1HPGDADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed