SCHEMBL6948973

SCHEMBL6948973

Nc1ncc2ncn(CCOc3ccccc3)c2n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.56
LTA4H P09960 4/20 0.53
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
ADRA1A P35348 1/20 0.48
HSD17B10 Q99714 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
LMNA P02545 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
HDAC6 Q9UBN7 1/20 0.44
TLR7 Q9NYK1 1/20 0.43
TP53 P04637 2/20 0.42
MAPT P10636 2/20 0.42
HTT P42858 1/20 0.42
HSP90AA1 P07900 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21596047 0.84 L3MBTL1 (0.56) L3MBTL1LTA4HNPC1RAB9AALDH1A1
SCHEMBL6950880 0.81 HTT (0.54) LTA4HKDM4EALDH1A1HPGDADRA1A
SCHEMBL2773942 0.80 ALDH1A1 (0.55) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL6361387 0.80 KDM4E (0.52) LTA4HKDM4EALDH1A1HPGDADRA1A
SCHEMBL6948072 0.78 ADORA2A (0.54) LTA4HKDM4EALDH1A1HPGDADRA1A
SCHEMBL3852270 0.78 KDM4E (0.50) LTA4HKDM4EALDH1A1HPGDADRA1A
SCHEMBL6946767 0.77 ADORA2A (0.50) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL28299548 0.77 HDAC6 (0.63) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL8933938 0.77 HSD17B10 (0.52) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL3151968 0.75 KDM4E (0.55) KDM4EALDH1A1HPGDADRA1AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed