SCHEMBL6947527

SCHEMBL6947527

O=CCc1ccc([N+](=O)[O-])c([N+](=O)[O-])c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.48
CYP3A4 P08684 1/20 0.48
CASP6 P55212 1/20 0.44
HTR1A P08908 1/20 0.42
DRD2 P14416 1/20 0.42
HTR2A P28223 1/20 0.42
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TDP1 Q9NUW8 2/20 0.38
MAPK1 P28482 1/20 0.38
ATM Q13315 1/20 0.38
ALDH5A1 P51649 1/20 0.38
ABAT P80404 1/20 0.38
VCAM1 P19320 1/20 0.38
SNCA P37840 1/20 0.38
POLB P06746 1/20 0.37
GPR35 Q9HC97 1/20 0.37
BACE1 P56817 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4313888 0.83 CYP19A1 (0.42) TSHRCYP3A4TDP1MAPK1ATM
SCHEMBL2772403 0.83 ALDH5A1 (0.59) TSHRMAPTNPSR1MAPK1ALDH5A1
SCHEMBL14893975 0.83 TDP1 (0.56) TSHRCYP3A4CASP6MAPTTDP1
SCHEMBL3903310 0.83 ALDH1A1 (0.45) CYP3A4MAPTNPSR1MAPK1ALDH5A1
SCHEMBL1983738 0.83 VCAM1 (0.59) TDP1VCAM1POLBALDH1A1
SCHEMBL9158 0.83 ALDH1A1 (0.55) MAPTNPSR1TDP1ATMVCAM1
SCHEMBL5716648 0.83 MAPT (0.50) TSHRCYP3A4MAPTTDP1POLB
SCHEMBL1225410 0.83 ALDH1A1 (0.53) TSHRCYP3A4MAPTNPSR1MAPK1
SCHEMBL4602487 0.80 PTGS2 (0.36) CYP3A4MAPTNPSR1TDP1MAPK1
SCHEMBL18138457 0.79 TSHR (0.52) TSHRCYP3A4CASP6HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230223-B1 OLIGOBENZIMIDAZOLE DERIVATIVES AND THEIR USE AS DNA TRANSFECTION AGENTS AVENTIS PHARMA SA (FR) 2004-02-25 EP disclosed
EP-1230223-A1 OLIGOBENZIMIDAZOLE DERIVATIVES AND THEIR USE AS DNA TRANSFECTION AGENTS Aventis Pharma S.A. (FR) 2002-08-14 EP disclosed
WO-2001032630-A1 OLIGOBENZIMIDAZOLE DERIVATIVES AND THEIR USE AS DNA TRANSFECTION AGENTS AVENTIS PHARMA S.A. (FR) 2001-05-10 WO disclosed