SCHEMBL6951247

SCHEMBL6951247

COC(=O)Oc1ccc2c(CCCCN3CCCC(Cc4ccc(C)cc4)C3)c[nH]c2c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.42
ACHE P22303 2/20 0.42
HTR2A P28223 1/20 0.41
CCR3 P51677 1/20 0.41
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
ADRA1D P25100 2/20 0.40
ADRA1A P35348 2/20 0.40
ADRA1B P35368 2/20 0.40
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959865 0.94 BCHE (0.49) BCHEACHEADRA2AADRA2BADRA2C
SCHEMBL6959528 0.93 CCR3 (0.46) HTR2ACCR3
SCHEMBL6955648 0.93 HTR2A (0.48) BCHEHTR2ACCR3
SCHEMBL7355747 0.92 BCHE (0.41) BCHEACHEHTR2ACCR3ADRA2A
SCHEMBL7075871 0.91 HTR1A (0.43) HTR2ACCR3
SCHEMBL6959392 0.88 ADRA2A (0.54) HTR2AADRA2AADRA2BADRA2CADRA1D
SCHEMBL7877114 0.88 NPC1 (0.49) BCHEACHEHTR2ACCR3ADRA2A
SCHEMBL6949399 0.88 ADRA2A (0.47) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL6954023 0.87 HTR1A (0.49) HTR2ACCR3ADRA2AADRA2BADRA2C
SCHEMBL6958383 0.87 HTR1A (0.52) BCHEACHEHTR2ACCR3ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP disclosed