SCHEMBL6954023

SCHEMBL6954023

COC(=O)Oc1ccc2[nH]cc(CCCCN3CCCC(Cc4ccc(F)cc4)C3)c2c1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.49
ADRA2A P08913 2/20 0.46
ADRA2B P18089 2/20 0.46
ADRA2C P18825 2/20 0.46
ADRA1D P25100 2/20 0.46
ADRA1A P35348 2/20 0.46
ADRA1B P35368 2/20 0.46
CCR3 P51677 3/20 0.46
CYP2D6 P10635 2/20 0.46
MPO P05164 1/20 0.46
HTR2A P28223 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959528 0.94 CCR3 (0.46) HTR1ACCR3CYP2D6HTR2A
SCHEMBL6959392 0.94 ADRA2A (0.54) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL6949399 0.93 ADRA2A (0.47) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL6959865 0.93 BCHE (0.49) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL6958383 0.92 HTR1A (0.52) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL7355825 0.91 MPO (0.48) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL7082018 0.90 HTR1A (0.48) HTR1A
SCHEMBL7880351 0.88 HTR1A (0.54) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL6951247 0.87 BCHE (0.42) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7350360 0.87 ADRA2A (0.54) HTR1AADRA2AADRA2BADRA2CADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP disclosed