SCHEMBL695593

SCHEMBL695593

CC(C)(C)OC(=O)N1C[C@H](S(=O)(=O)CC2CC2)C[C@H]1C(=O)N(C#N)C1CC1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
NR1H2 P55055 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CTSS P25774 5/20 0.33
CTSL P07711 3/20 0.33
CTSB P07858 2/20 0.33
CTSK P43235 2/20 0.33
UCHL1 P09936 1/20 0.31
USP30 Q70CQ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL695975 0.87 CTSL (0.34) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL700342 0.81 SMN1; SMN2 (0.43) KMT2ANR1H2SMN1; SMN2CTSSCTSL
SCHEMBL15200625 0.80 CYP1A2 (0.43) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL695599 0.80 CYP1A2 (0.43) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL696865 0.79 CTSS (0.41) CTSSCTSLCTSBCTSKUCHL1
SCHEMBL699042 0.79 NR1H2 (0.39) ALDH1A1KMT2ANR1H2SMN1; SMN2CTSS
SCHEMBL696541 0.78 UCHL1 (0.37) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL694346 0.78 STS (0.44) CTSSCTSLCTSBCTSKUCHL1
SCHEMBL15202523 0.78 STS (0.44) MEN1KMT2ACTSSCTSLCTSB
SCHEMBL695674 0.78 CTSS (0.40) CTSSCTSLCTSBCTSKUCHL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed