SCHEMBL6957839

SCHEMBL6957839

Cc1cc(C)cc(Sc2nc(C(C)O)[nH]c2C(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
ALDH1A1 P00352 1/20 0.33
ALOX15 P16050 1/20 0.33
MEN1 O00255 1/20 0.30
HTT P42858 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973698 0.86 GPR84 (0.30)
SCHEMBL6965300 0.84 CYP1A2 (0.33) CYP1A2ALDH1A1ALOX15MEN1KMT2A
SCHEMBL6973960 0.81 IDO1 (0.38) ALDH1A1HTTKMT2A
SCHEMBL6961420 0.81 DHFR (0.36) CYP1A2ALDH1A1ALOX15MEN1HTT
SCHEMBL6973795 0.80 GSK3B (0.32) CYP1A2MEN1KMT2A
SCHEMBL6961917 0.77 HAO1 (0.38) CYP1A2ALDH1A1ALOX15MEN1KMT2A
SCHEMBL6972114 0.77 LMNA (0.41) CYP1A2ALDH1A1MEN1KMT2A
SCHEMBL7086346 0.77 CYP1A2 (0.40) CYP1A2ALDH1A1ALOX15MEN1HTT
SCHEMBL7084364 0.72 HSP90B1 (0.32)
SCHEMBL6967234 0.71 TYMS (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed