SCHEMBL6973960

SCHEMBL6973960

Cc1cc(C)cc(Sc2nc(C(O)Cc3ccccc3)[nH]c2C(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.38
TRPA1 O75762 2/20 0.37
ADRB2 P07550 4/20 0.33
LMNA P02545 2/20 0.32
MAPT P10636 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
ALPL P05186 1/20 0.32
ALPI P09923 1/20 0.32
ALPG P10696 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TACR1 P25103 2/20 0.32
TAAR1 Q96RJ0 2/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31
SLC18A2 Q05940 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973795 0.90 GSK3B (0.32) KMT2APOLB
SCHEMBL7081023 0.87 TRPA1 (0.33) IDO1TRPA1ADRB2LMNATAAR1
SCHEMBL6973698 0.84 GPR84 (0.30)
SCHEMBL6973409 0.82 SLC6A4 (0.36) TRPA1KMT2ASLC6A4ALDH1A1
SCHEMBL6967546 0.81 IDO1 (0.38) IDO1TRPA1ADRB2LMNAMAPT
SCHEMBL6957839 0.81 CYP1A2 (0.40) HTTKMT2AALDH1A1
SCHEMBL6968179 0.77 CYP1A2 (0.33)
SCHEMBL6974054 0.77 GSK3B (0.32)
SCHEMBL6974320 0.75 MAPK14 (0.34) SMN1; SMN2
SCHEMBL7082933 0.75 CSNK2A2 (0.38) LMNAMAPTSMN1; SMN2KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed