SCHEMBL6973795

SCHEMBL6973795

Cc1cc(C)cc(Sc2nc(C(O)Cc3ccncc3)[nH]c2C(C)C)c1

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.32
CDC7 O00311 1/20 0.32
GAA P10253 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
POLB P06746 1/20 0.31
MAPK14 Q16539 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973960 0.90 IDO1 (0.38) POLBKMT2A
SCHEMBL6968179 0.88 CYP1A2 (0.33) GSK3BCDC7CYP1A2CYP3A4CYP2C9
SCHEMBL6974054 0.88 GSK3B (0.32) GSK3BCDC7CYP1A2CYP3A4CYP2C9
SCHEMBL6973409 0.86 SLC6A4 (0.36) GAACDK5CDK5R1CYP1A2CYP3A4
SCHEMBL6973698 0.83 GPR84 (0.30)
SCHEMBL7082933 0.83 CSNK2A2 (0.38) GAACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6974320 0.83 MAPK14 (0.34) CYP3A4MAPK14
SCHEMBL7083004 0.82 GSK3B (0.32) GSK3BGAACYP1A2CYP3A4CYP2C9
SCHEMBL6957839 0.80 CYP1A2 (0.40) CYP1A2MEN1KMT2A
SCHEMBL6968078 0.79 ALOX5 (0.38) CDC7CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed