SCHEMBL6958300

SCHEMBL6958300

CSc1sc(OC(=O)O)cc1Br

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33
TSHR P16473 1/20 0.30
HSD17B10 Q99714 1/20 0.30
TPMT P51580 1/20 0.30
PKM P14618 1/20 0.30
LIG1 P18858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201000 0.76 GSK3B (0.41) PKM
SCHEMBL6924925 0.73 KEAP1 (0.57) KEAP1NFE2L2LCKFYNPKM
SCHEMBL9158487 0.73 DAO (0.34)
SCHEMBL6970016 0.72 ALDH1A1 (0.41)
SCHEMBL6923952 0.69 KEAP1 (0.41) KEAP1NFE2L2TSHRHSD17B10PKM
SCHEMBL5046977 0.66 GPR35 (0.33)
SCHEMBL9176677 0.66 MAPT (0.52) HSD17B10
SCHEMBL5200748 0.64 CHRNA1 (0.39) HSD17B10
SCHEMBL5202302 0.63 SLC9A1 (0.48)
SCHEMBL10882465 0.63 DAO (0.55) TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676395-B1 Substituted N-heteroaroylguanidines, as inhibitors of sodium-hydrogen exchange, as antiarrhythmic agents and as inhibitors of the proliferation of cells HOECHST AG (DE) 2003-09-03 EP disclosed
EP-0676395-A2 Substituted N-heteroaroylguanidines, as inhibitors of sodium-hydrogen exchange, as antiarrhythmic agents and as inhibitors of the proliferation of cells HOECHST AKTIENGESELLSCHAFT (DE) 1995-10-11 EP disclosed