SCHEMBL6958744

SCHEMBL6958744

CCOC(=O)CN1C(=O)CC(C)N(C(=O)c2ccc(N)cc2)c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
NPSR1 Q6W5P4 1/20 0.47
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
PPARG P37231 1/20 0.42
LMNA P02545 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 1/20 0.40
GAA P10253 2/20 0.39
RAB9A P51151 1/20 0.39
MCL1 Q07820 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
USP2 O75604 1/20 0.38
HTT P42858 1/20 0.38
MAPT P10636 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAOA P21397 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972297 0.86 ALDH1A1 (0.46) ALDH1A1NPSR1MEN1KMT2APPARG
SCHEMBL6960127 0.79 NPSR1 (0.49) ALDH1A1NPSR1MEN1KMT2APPARG
SCHEMBL6972433 0.79 AVPR2 (0.54) ALDH1A1MAPT
SCHEMBL6973134 0.78 NPSR1 (0.47) ALDH1A1NPSR1MEN1KMT2APPARG
SCHEMBL6969459 0.71 ALDH1A1 (0.46) ALDH1A1NPSR1MEN1KMT2APPARG
SCHEMBL6969797 0.70 LMNA (0.44) ALDH1A1NPSR1MEN1KMT2APPARG
SCHEMBL6959586 0.69 HDAC1 (0.49) NPSR1CYP3A4
SCHEMBL6972107 0.69 NOTUM (0.46) ALDH1A1NPSR1MEN1KMT2ALMNA
SCHEMBL6970661 0.69 ALDH1A1 (0.46) ALDH1A1NPSR1MEN1KMT2APPARG
SCHEMBL6967260 0.68 AVPR2 (0.48) ALDH1A1MEN1KMT2ALMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed