SCHEMBL6959586

SCHEMBL6959586

CC(C)(C)OC(=O)CN1C(=O)CN(C(=O)c2ccc(N)cc2)c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
AVPR2 P30518 1/20 0.40
AVPR1A P37288 1/20 0.40
KCNN4 O15554 1/20 0.37
KCNA3 P22001 1/20 0.37
CCKBR P32239 2/20 0.37
XIAP P98170 2/20 0.37
P2RX4 Q99571 1/20 0.36
CYP3A4 P08684 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959376 0.85 HDAC1 (0.46) HDAC1HDAC6XIAPP2RX4
SCHEMBL6967260 0.77 AVPR2 (0.48) AVPR2AVPR1AXIAPCYP3A4
SCHEMBL6959609 0.77 AVPR2 (0.50) AVPR2AVPR1A
SCHEMBL6959648 0.76 AVPR1A (0.42) HDAC1HDAC6AVPR2AVPR1AKCNN4
SCHEMBL6960127 0.75 NPSR1 (0.49) AVPR2AVPR1ACYP3A4NPSR1
SCHEMBL6970428 0.75 CYP2D6 (0.43) AVPR2AVPR1AKCNN4KCNA3NPSR1
SCHEMBL6967996 0.72 AVPR2 (0.47) AVPR2AVPR1ACYP3A4
SCHEMBL5966758 0.71 CCKBR (0.48) CCKBR
SCHEMBL6958744 0.69 ALDH1A1 (0.49) CYP3A4NPSR1
SCHEMBL29286990 0.69 MEN1 (0.48) NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed