SCHEMBL6959588

SCHEMBL6959588

Cc1ccc(-c2ccccc2C(=O)Nc2ncccc2C(=O)O)cc1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.61
L3MBTL1 Q9Y468 2/20 0.61
CHRNB2 P17787 3/20 0.54
CHRNB4 P30926 3/20 0.54
CHRNA3 P32297 3/20 0.54
CHRNA4 P43681 3/20 0.54
DHODH Q02127 4/20 0.49
GAA P10253 4/20 0.49
LMNA P02545 1/20 0.49
ALDH1A1 P00352 2/20 0.49
HTT P42858 1/20 0.48
KDM4E B2RXH2 1/20 0.48
SORT1 Q99523 1/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
MEN1 O00255 2/20 0.46
MAPT P10636 1/20 0.46
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18640758 0.82 NPC1 (0.61) KMT2AL3MBTL1DHODHGAALMNA
SCHEMBL8800517 0.81 KMT2A (0.67) KMT2AL3MBTL1DHODHGAALMNA
SCHEMBL7568546 0.80 CHRNB2 (0.62) KMT2AL3MBTL1CHRNB2CHRNB4CHRNA3
Toluene SCHEMBL8797778 0.78 DHODH (0.56) KMT2AL3MBTL1DHODHGAALMNA
Toluene SCHEMBL8650718 0.78 DHODH (0.56) KMT2AL3MBTL1DHODHGAALMNA
SCHEMBL14398931 0.78 DHODH (0.56) KMT2AL3MBTL1DHODHGAALMNA
SCHEMBL31393753 0.78 CHRNB2 (0.78) KMT2AL3MBTL1CHRNB2CHRNB4CHRNA3
SCHEMBL6959593 0.78 ALDH1A1 (0.53) KMT2AL3MBTL1CHRNB2CHRNB4CHRNA3
SCHEMBL18640842 0.77 KMT2A (0.64) KMT2ADHODHGAAALDH1A1HTT
SCHEMBL372 0.77 KMT2A (0.60) KMT2AGAAALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed