SCHEMBL6960079

SCHEMBL6960079

O=C1c2ccccc2C(=O)N1CCCCCCN1C(=O)CCN(C(=O)c2ccc([N+](=O)[O-])cc2)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
NPSR1 Q6W5P4 3/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
CYP2D6 P10635 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
DRD2 P14416 2/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
TSHR P16473 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HTR1A P08908 2/20 0.42
MAPK1 P28482 1/20 0.42
HTR2A P28223 1/20 0.41
HTR7 P34969 1/20 0.41
HTR6 P50406 1/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971119 0.89 DRD2 (0.46) ALDH1A1NPSR1CYP3A4CYP2C9CYP2C19
SCHEMBL6964588 0.86 AVPR2 (0.46) ALDH1A1CYP3A4CYP2D6SMN1; SMN2DRD2
SCHEMBL6958687 0.84 DRD3 (0.46) ALDH1A1CYP2D6DRD2DRD4DRD3
SCHEMBL6955542 0.82 ALDH1A1 (0.43) ALDH1A1DRD2DRD4DRD3TSHR
SCHEMBL6969761 0.81 L3MBTL1 (0.43) ALDH1A1SMN1; SMN2DRD2DRD4DRD3
SCHEMBL6969126 0.79 L3MBTL1 (0.45) ALDH1A1SMN1; SMN2DRD2DRD4DRD3
SCHEMBL7140109 0.78 L3MBTL1 (0.45) ALDH1A1SMN1; SMN2L3MBTL1HTR1AHPGD
SCHEMBL6955643 0.77 L3MBTL1 (0.46) ALDH1A1NPSR1SMN1; SMN2L3MBTL1MEN1
SCHEMBL7352575 0.76 ALDH1A1 (0.56) ALDH1A1TSHRL3MBTL1HPGD
SCHEMBL6961373 0.75 AVPR2 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed