SCHEMBL6971119

SCHEMBL6971119

O=C1CCN(C(=O)c2ccc([N+](=O)[O-])cc2)c2ccccc2N1CCCCCCCl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.46
DRD4 P21917 2/20 0.46
DRD3 P35462 2/20 0.46
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
BCHE P06276 1/20 0.40
P2RX4 Q99571 1/20 0.40
STING1 Q86WV6 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960079 0.89 ALDH1A1 (0.48) DRD2DRD4DRD3GRIN1GRIN2B
SCHEMBL6958687 0.85 DRD3 (0.46) DRD2DRD4DRD3GRIN1GRIN2B
SCHEMBL6955542 0.83 ALDH1A1 (0.43) DRD2DRD4DRD3L3MBTL1NPC1
SCHEMBL6969761 0.82 L3MBTL1 (0.43) DRD2DRD4DRD3GRIN1GRIN2B
SCHEMBL6969126 0.80 L3MBTL1 (0.45) DRD2DRD4DRD3L3MBTL1NPC1
SCHEMBL7140109 0.79 L3MBTL1 (0.45) L3MBTL1NPC1RAB9AHPGDALDH1A1
SCHEMBL6955643 0.77 L3MBTL1 (0.46) L3MBTL1NPC1RAB9AHPGDALDH1A1
SCHEMBL6964416 0.76 DRD2 (0.50) DRD2DRD4DRD3GRIN1GRIN2B
SCHEMBL6970758 0.76 ALDH1A1 (0.45) L3MBTL1HTTALDH1A1MAPT
SCHEMBL6969043 0.75 DRD3 (0.47) DRD2DRD4DRD3L3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed