SCHEMBL696072

SCHEMBL696072

COC(=O)C1CCCN1C(=O)CC(=O)CS(=O)(=O)c1ccc(F)cc1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.42
HSD11B1 P28845 2/20 0.41
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.39
PEPD P12955 1/20 0.39
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PDK2 Q15119 1/20 0.38
KLK5 Q9Y337 1/20 0.38
ACE P12821 1/20 0.38
P2RX7 Q99572 2/20 0.37
LOX P28300 1/20 0.37
PKM P14618 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CG P48736 1/20 0.36
FKBP1A P62942 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL695737 0.91 ALDH1A1 (0.51) ALDH1A1GAAPEPDLMNARAB9A
SCHEMBL696406 0.87 ALDH1A1 (0.48) EPHX2ALDH1A1GAALMNARAB9A
SCHEMBL696794 0.77 ALDH1A1 (0.48) ALDH1A1LMNARAB9ASMN1; SMN2KLK5
SCHEMBL695502 0.76 ACE (0.48) HSD11B1ALDH1A1LMNARAB9ASMN1; SMN2
SCHEMBL695669 0.73 POLB (0.46) ALDH1A1PEPDLMNARAB9ASMN1; SMN2
SCHEMBL696071 0.71 CTSS (0.43) EPHX2HSD11B1P2RX7
SCHEMBL2105751 0.71 CTSS (0.43) EPHX2HSD11B1P2RX7
SCHEMBL30546762 0.69 P2RX7 (0.61) ALDH1A1GAASMN1; SMN2P2RX7PKM
SCHEMBL30546740 0.69 P2RX7 (0.61) ALDH1A1GAASMN1; SMN2P2RX7PKM
SCHEMBL697248 0.69 LMNA (0.45) ALDH1A1PEPDLMNARAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed