SCHEMBL6960840

SCHEMBL6960840

CCn1ncc(-c2ccc3c(c2)c(C2=CCNCC2)cn3-c2ccc(F)cc2)n1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.51
HTR1B P28222 2/20 0.51
HTR6 P50406 8/20 0.46
KHK P50053 2/20 0.44
KCNH2 Q12809 1/20 0.39
DRD2 P14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6962346 0.89 HTR1A (0.50) HTR1AHTR1BHTR6KHKKCNH2
SCHEMBL6962241 0.81 DRD2 (0.49) HTR1AHTR1BHTR6KHKKCNH2
SCHEMBL9462735 0.80 HTR6 (0.68) HTR1AHTR6KHKKCNH2
SCHEMBL6954562 0.79 DRD2 (0.56) HTR1AHTR1BHTR6KHKKCNH2
SCHEMBL6966491 0.79 HTR1A (0.69) HTR1AHTR1BKCNH2DRD2
SCHEMBL6580736 0.76 HTR6 (0.61) HTR1AHTR6KCNH2DRD2
Hydrochloric Acid SCHEMBL27751697 0.76 HTR6 (0.61) HTR1AHTR6KCNH2DRD2
SCHEMBL9462566 0.75 HTR6 (0.56) HTR1AHTR6KCNH2
SCHEMBL6583508 0.75 HTR6 (0.54) HTR1AHTR6KHKKCNH2
SCHEMBL6955047 0.74 DRD2 (0.52) HTR1AHTR6KHKKCNH2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602889-B1 5-heteroaryl substituted indoles H. LUNDBECK A.S. (DK) 2003-08-05 US disclosed
EP-1068198-B1 5-HETEROARYL SUBSTITUTED INDOLES LUNDBECK & CO AS H (DK) 2003-05-28 EP disclosed