SCHEMBL6961376

SCHEMBL6961376

NNc1ccccc1-c1ccsc1C(N)=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.58
MAPK8 P45983 2/20 0.44
MAPK10 P53779 1/20 0.44
ACHE P22303 1/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
PKM P14618 1/20 0.37
RORC P51449 1/20 0.36
RORB Q92753 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
HTR2B P41595 1/20 0.36
IKBKB O14920 2/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPT P10636 2/20 0.34
HTR1A P08908 1/20 0.34
HTR7 P34969 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4717953 0.78 BCAT2 (0.64) BCAT2MAPK8MAPK10ALDH1A1KDM4E
SCHEMBL12495840 0.77 BCAT2 (0.62) BCAT2MAPK8MAPK10ALDH1A1KDM4E
SCHEMBL7472100 0.77 BCAT2 (0.62) BCAT2MAPK8MAPK10PKMRORC
SCHEMBL27576830 0.74 BCAT2 (0.58) BCAT2MAPK8MAPK10ALDH1A1KDM4E
SCHEMBL4445671 0.74 BCAT2 (1.00) BCAT2MAPK8MAPK10ALDH1A1RORB
SCHEMBL28012573 0.73 BCAT2 (0.57) BCAT2MAPK8ALDH1A1KDM4EPOLB
Hydrochloric Acid SCHEMBL31228833 0.73 BCAT2 (0.96) BCAT2MAPK8MAPK10ALDH1A1RORB
SCHEMBL11817898 0.72 ALDH1A1 (0.46) ALDH1A1KDM4EPOLBPKMMEN1
SCHEMBL31661830 0.69 MKNK1 (0.54) BCAT2ALDH1A1KDM4EPOLBIRAK4
SCHEMBL10798532 0.69 RORB (0.40) BCAT2MAPK8MAPK10ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed