SCHEMBL6961885

SCHEMBL6961885

CCn1c(CO)nc(C(C)C)c1Sc1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
GRM5 P41594 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
DHODH Q02127 4/20 0.34
POLB P06746 1/20 0.34
AKR1B1 P15121 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960470 0.91 TP53 (0.36) TP53RXFP1GRM5MEN1KMT2A
SCHEMBL6965320 0.91 MEN1 (0.36) TP53RXFP1GRM5MEN1KMT2A
SCHEMBL6971946 0.89 TLR8 (0.40) TP53RXFP1GRM5MEN1KMT2A
SCHEMBL6966003 0.88 TYMS (0.37) TP53RXFP1GRM5MEN1KMT2A
SCHEMBL6160601 0.88 HSP90B1 (0.33) DHODH
SCHEMBL6975192 0.88 TDP1 (0.43) TP53RXFP1MEN1KMT2ANPSR1
SCHEMBL6966933 0.87 TSHR (0.35) TP53RXFP1GRM5MEN1KMT2A
SCHEMBL7080431 0.86 MEN1 (0.36) TP53RXFP1GRM5MEN1KMT2A
SCHEMBL6963544 0.86 POLB (0.45) TP53RXFP1GRM5MEN1KMT2A
SCHEMBL7087601 0.86 SLC6A9 (0.33) TP53RXFP1GRM5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed