SCHEMBL6966933

SCHEMBL6966933

C=CCn1c(CO)nc(C(C)C)c1Sc1cccc(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.35
RECQL P46063 1/20 0.35
TP53 P04637 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
MAPT P10636 2/20 0.35
GAA P10253 1/20 0.35
PPARG P37231 1/20 0.35
HTT P42858 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HSD17B10 Q99714 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
LMNA P02545 1/20 0.34
GRM5 P41594 3/20 0.34
L3MBTL1 Q9Y468 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973144 0.90 TSHR (0.35) TSHRRECQLTP53NPSR1MAPT
SCHEMBL6965321 0.89 APLNR (0.34) TP53NPSR1MAPTGAAPPARG
SCHEMBL6961885 0.87 TP53 (0.37) TP53NPSR1LMNAGRM5L3MBTL1
SCHEMBL6965320 0.85 MEN1 (0.36) TP53NPSR1MAPTHTTALDH1A1
SCHEMBL6975192 0.84 TDP1 (0.43) TP53NPSR1ALDH1A1HPGDKDM4E
SCHEMBL6970754 0.83 TDP1 (0.34) TSHRRECQLTP53NPSR1MAPT
SCHEMBL6976452 0.83 CFTR (0.40) MAPTALDH1A1HPGDAPOBEC3GLMNA
SCHEMBL7079909 0.82 IDO1 (0.36) TP53NPSR1ALDH1A1HPGDKDM4E
SCHEMBL6969476 0.82 MEN1 (0.39) TP53NPSR1MAPTGAAALDH1A1
SCHEMBL6969810 0.81 APLNR (0.35) TSHRMAPTGAAALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed