SCHEMBL6975192

SCHEMBL6975192

CC(C)c1nc(CO)n(Cc2ccccc2)c1Sc1cccc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.43
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TP53 P04637 4/20 0.38
RXFP1 Q9HBX9 1/20 0.37
LMNA P02545 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CCR2 P41597 1/20 0.36
KCNJ6 P48051 1/20 0.36
KCNJ5 P48544 1/20 0.36
KCNJ3 P48549 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
SLC6A9 P48067 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7079909 0.92 IDO1 (0.36) TDP1MEN1KMT2ANPSR1L3MBTL1
SCHEMBL6966848 0.91 TDP1 (0.42) TDP1MEN1KMT2ATP53KCNJ6
SCHEMBL6970034 0.90 ALDH1A1 (0.40) TDP1KMT2ATP53LMNAKDM4E
SCHEMBL6961885 0.88 TP53 (0.37) TDP1MEN1KMT2ANPSR1L3MBTL1
SCHEMBL7079929 0.87 GRM5 (0.38) TDP1MEN1KMT2ANPSR1L3MBTL1
SCHEMBL6974703 0.86 TDP1 (0.41) TDP1MEN1KMT2ANPSR1L3MBTL1
SCHEMBL6965320 0.86 MEN1 (0.36) TDP1MEN1KMT2ANPSR1L3MBTL1
Acetamide SCHEMBL6972197 0.85 TDP1 (0.41) TDP1MEN1KMT2ANPSR1L3MBTL1
SCHEMBL6967543 0.84 TDP1 (0.38) TDP1MEN1KMT2AL3MBTL1TP53
SCHEMBL6966621 0.84 TDP1 (0.40) TDP1MEN1KMT2ANPSR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed