SCHEMBL6962491

SCHEMBL6962491

O=Cc1ccc(O)c(NC(=O)CCl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.47
KDM4E B2RXH2 3/20 0.47
RAB9A P51151 2/20 0.47
PTGS2 P35354 1/20 0.47
ALDH1A1 P00352 7/20 0.44
HTT P42858 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
HPGD P15428 2/20 0.43
HDAC1 Q13547 1/20 0.41
MAPK1 P28482 2/20 0.41
NPC1 O15118 1/20 0.41
MITF O75030 1/20 0.41
THRB P10828 1/20 0.41
ALOX15 P16050 1/20 0.40
ALDH5A1 P51649 2/20 0.40
ABAT P80404 2/20 0.40
GAA P10253 2/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967818 0.87 ALDH1A1 (0.47) POLBKDM4ERAB9APTGS2ALDH1A1
SCHEMBL3755148 0.80 POLB (0.53) POLBKDM4ERAB9AALDH1A1HTT
SCHEMBL29914686 0.80 POLB (0.53) POLBKDM4ERAB9AALDH1A1HTT
SCHEMBL10029204 0.79 ALDH1A1 (0.67) KDM4ERAB9AALDH1A1HTTSMN1; SMN2
SCHEMBL7684154 0.78 KDM4E (0.54) POLBKDM4ERAB9APTGS2ALDH1A1
SCHEMBL21409465 0.78 MITF (0.51) POLBKDM4ERAB9AALDH1A1HTT
SCHEMBL29957610 0.78 KDM4E (0.54) POLBKDM4ERAB9APTGS2ALDH1A1
SCHEMBL247350 0.78 POLB (0.75) POLBMEN1KMT2AHPGDMAPK1
SCHEMBL30612630 0.78 POLB (0.75) POLBMEN1KMT2AHPGDMAPK1
SCHEMBL16858580 0.77 POLB (0.50) POLBKDM4ERAB9AALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906294-B1 BENZOXAZINONE DOPAMINE D4 RECEPTOR ANTAGONISTS WARNER LAMBERT CO (US) 2003-01-29 EP disclosed
US-6177422-B1 ANTIPSYCHOTIC AGENT WITH REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0906294-A1 BENZOXAZINONE DOPAMINE D4 RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1999-04-07 EP disclosed
WO-1997045419-A1 BENZOXAZINONE DOPAMINE D4 RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1997-12-04 WO disclosed