SCHEMBL6962874

SCHEMBL6962874

COc1cccc(SC(C(=O)O)C(=O)O)c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 13/20 0.56
MTNR1B P49286 13/20 0.56
ALDH1A1 P00352 1/20 0.48
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
EDNRA P25101 2/20 0.47
LMNA P02545 1/20 0.46
PARP1 P09874 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7371129 0.81 MTNR1B (0.54) MTNR1AMTNR1BALDH1A1
SCHEMBL5304699 0.80 MTNR1A (0.56) MTNR1AMTNR1BALDH1A1CES2CES1
SCHEMBL5992093 0.78 MTNR1A (0.57) MTNR1AMTNR1BALDH1A1CES2CES1
SCHEMBL6960077 0.77 KIF11 (0.40) LMNAPARP1
SCHEMBL10297508 0.77 MTNR1A (0.55) MTNR1AMTNR1BALDH1A1
SCHEMBL10702424 0.75 MAPT (0.55) MTNR1AMTNR1BALDH1A1LMNA
SCHEMBL10426256 0.75 MTNR1A (0.51) MTNR1AMTNR1BLMNA
SCHEMBL7461488 0.75 MTNR1A (0.54) MTNR1AMTNR1BALDH1A1
SCHEMBL28470846 0.74 MTNR1A (0.55) MTNR1AMTNR1BCES2CES1EDNRA
SCHEMBL6958711 0.74 CYP2C9 (0.43) ALDH1A1LMNAPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729465-B1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & CO (US) 2003-01-22 EP disclosed
US-6005103-A TREATMENT OF BACTERIAL AND VIRAL INFECTIONS AND DISEASES, INCLUDING AIDS WARNER-LAMBERT COMPANY (US) 1999-12-21 US disclosed
US-5808062-A AIDS THERAPY WARNER-LAMBERT COMPANY (US) 1998-09-15 US disclosed