SCHEMBL6963124

SCHEMBL6963124

CCNc1cc(Sc2cccc3cnccc23)c(Cl)cc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
IMPDH2 P12268 1/20 0.36
TRPV1 Q8NER1 5/20 0.36
CCR4 P51679 1/20 0.35
AOC1 P19801 1/20 0.34
AOC3 Q16853 1/20 0.34
ALDH1A1 P00352 4/20 0.34
ROCK2 O75116 4/20 0.34
HTT P42858 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
ROCK1 Q13464 2/20 0.34
HPGD P15428 2/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6962927 0.84 LMNA (0.51) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6965142 0.72 PDE7A (0.47) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6968741 0.72 KDM4E (0.57) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6968806 0.71 LMNA (0.51) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL11142216 0.71 ALDH1A1 (0.53) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6973375 0.71 LMNA (0.54) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6974563 0.70 KDM4E (0.41) LMNAALDH1A1HTTSMN1; SMN2L3MBTL1
SCHEMBL6966199 0.69 HDAC6 (0.42) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6973379 0.69 CYP3A4 (0.51) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6963171 0.68 AR (0.53) LMNACYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed