SCHEMBL6963346

SCHEMBL6963346

C=CCOC(=O)N1C[C@@H](N2CC[C@H](Br)C2=O)C[C@H]1C(=O)N(C)C

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.33
CYP19A1 P11511 1/20 0.32
FAAH O00519 3/20 0.31
MGLL Q99685 1/20 0.31
CHRM1 P11229 1/20 0.31
ELANE P08246 1/20 0.30
CTSG P08311 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6954836 1.00 SIGMAR1 (0.33) SIGMAR1CYP19A1FAAHMGLLCHRM1
Bromide SCHEMBL6958973 0.81 FAAH (0.38) SIGMAR1CYP19A1FAAHMGLLCHRM1
Bromide SCHEMBL6958976 0.81 FAAH (0.38) SIGMAR1CYP19A1FAAHMGLLCHRM1
Bromide SCHEMBL6963355 0.77 SIGMAR1 (0.33) SIGMAR1CYP19A1FAAHMGLLCHRM1
SCHEMBL6956392 0.77 CHRM1 (0.34) SIGMAR1FAAHMGLLCHRM1
SCHEMBL6965750 0.77 ERN1 (0.35) FAAHMGLLCHRM1
SCHEMBL6772112 0.75 POLB (0.36) SIGMAR1CYP19A1
SCHEMBL6968586 0.74 L3MBTL1 (0.36) FAAHMGLLCHRM1
SCHEMBL6970169 0.74 L3MBTL1 (0.36) FAAHMGLLCHRM1
SCHEMBL6970899 0.74 L3MBTL1 (0.36) FAAHMGLLCHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0849269-B9 Vinyl pyrrolidine cephalosporins with basic substituents BASILEA PHARMACEUTICA AG (CH) 2003-03-05 EP disclosed
EP-0849269-B1 Vinyl pyrrolidine cephalosporins with basic substituents BASILEA PHARMACEUTICA AG (CH) 2002-07-10 EP disclosed
US-5981519-A Vinyl-pyrrolidinone cephalosporins HOFFMAN-LA ROCHE INC. (US) 1999-11-09 US disclosed
EP-0849269-A1 Vinyl pyrrolidine cephalosporins with basic substituents F. HOFFMANN-LA ROCHE AG (CH) 1998-06-24 EP disclosed