SCHEMBL6963394

SCHEMBL6963394

O=c1[nH]c2cc([S+]([O-])c3cccc4cnccc34)c([N+](=O)[O-])cc2s1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PGR P06401 2/20 0.39
PDE3B Q13370 4/20 0.36
PDE3A Q14432 4/20 0.36
CHUK O15111 1/20 0.35
PKN1 Q16512 1/20 0.32
PKN2 Q16513 1/20 0.32
SYK P43405 1/20 0.32
MAPT P10636 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
PIM1 P11309 1/20 0.30
PIM3 Q86V86 1/20 0.30
HIPK2 Q9H2X6 1/20 0.30
DAO P14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970313 0.79 PGR (0.39) PGRPDE3BPDE3ACHUKPKN1
SCHEMBL1010663 0.66 ALDH1A1 (0.61) PKN1PKN2MAPTALDH1A1LMNA
SCHEMBL29674805 0.66 ALDH1A1 (0.61) PKN1PKN2MAPTALDH1A1LMNA
SCHEMBL27415737 0.65 ALDH1A1 (0.59) PKN1PKN2MAPTALDH1A1LMNA
Methane SCHEMBL27506999 0.65 ALDH1A1 (0.59) PKN1PKN2MAPTALDH1A1LMNA
Bromide SCHEMBL11820178 0.65 ALDH1A1 (0.59) PKN1PKN2MAPTALDH1A1LMNA
SCHEMBL8355731 0.65 CYP3A4 (0.35) MAPTLMNA
Nitric Acid SCHEMBL6691619 0.63 ALDH1A1 (0.56) PKN1PKN2MAPTALDH1A1LMNA
SCHEMBL6963305 0.63 CMA1 (0.47) PGRMAPTALDH1A1LMNA
SCHEMBL11110839 0.63 PGR (0.47) PGRPDE3BPDE3AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed