SCHEMBL7084495

SCHEMBL7084495

CC(=O)OC(Cc1ccccn1)c1nc(C(C)C)c(Sc2ccccc2)[nH]1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRA P18433 1/20 0.37
CYP1A2 P05177 3/20 0.34
TSHR P16473 2/20 0.34
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ALDH1A1 P00352 2/20 0.33
PGR P06401 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
PTGS1 P23219 1/20 0.32
SLC6A2 P23975 1/20 0.32
FDPS P14324 1/20 0.32
MAOB P27338 1/20 0.32
FNTA P49354 2/20 0.32
FNTB P49356 2/20 0.32
KMT2A Q03164 1/20 0.31
HTT P42858 1/20 0.31
ATM Q13315 1/20 0.31
NPC1 O15118 1/20 0.31
TUBB4A P04350 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7081154 0.90 MAPT (0.35) PTPRAMAPTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL7084827 0.90 SLC6A9 (0.34) PTPRAALDH1A1KMT2A
SCHEMBL7078977 0.90 RHEB (0.34) PTPRACYP1A2TSHRMAPTALDH1A1
SCHEMBL6973462 0.90 ALDH1A1 (0.32) PTPRACYP1A2TSHRALDH1A1PGR
SCHEMBL7080029 0.88 PTPRA (0.34) PTPRACYP1A2TSHRCYP2D6MAPT
SCHEMBL7084594 0.87 CYP1A2 (0.38) CYP1A2MAPTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL6975056 0.86 ALDH1A1 (0.36) ALDH1A1FNTAFNTBTUBB4ATUBB
SCHEMBL6974480 0.84 DHFR (0.34) ALDH1A1KMT2ATUBB4ATUBBTUBA3C
SCHEMBL6974559 0.84 PTPRA (0.32) PTPRAFDPSDHFR
SCHEMBL6969311 0.83 LMNA (0.37) CYP1A2SMN1; SMN2FDPSFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed