SCHEMBL6964520

SCHEMBL6964520

COc1ccc(COCc2nc(C(C)C)c(Sc3cc(Cl)cc(Cl)c3)n2C)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.34
TRPV6 Q9H1D0 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
TBXAS1 P24557 2/20 0.32
CYP3A4 P08684 2/20 0.32
MAPT P10636 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
TP53 P04637 1/20 0.31
GAA P10253 1/20 0.31
PTGIR P43119 1/20 0.31
IDO1 P14902 1/20 0.31
DHFR P00374 1/20 0.31
CCR2 P41597 1/20 0.31
DCTPP1 Q9H773 1/20 0.31
NPBWR1 P48145 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6966985 0.91 MAPT (0.35) DHODHCYP3A4MAPTSMN1; SMN2TP53
SCHEMBL6974846 0.89 MEN1 (0.36) DHODHTRPV6CA1CA2TBXAS1
SCHEMBL6969238 0.89 VCP (0.38) DHODHHRH4SMN1; SMN2KDM4ERAB9A
SCHEMBL6965629 0.88 DHFR (0.33) DHODHTRPV6HRH4MAPTSMN1; SMN2
SCHEMBL6974229 0.88 MAPT (0.34) DHODHCA1CA2TBXAS1CYP3A4
SCHEMBL14439857 0.85 DHODH (0.39) DHODHMAPTSMN1; SMN2TP53GAA
SCHEMBL6957630 0.85 DHODH (0.39) DHODHMAPTSMN1; SMN2TP53GAA
SCHEMBL6967218 0.85 MAPT (0.35) DHODHTBXAS1MAPTSMN1; SMN2TP53
SCHEMBL6963914 0.85 NPC1 (0.38) DHODHCYP3A4MAPTSMN1; SMN2TP53
SCHEMBL6958208 0.85 MAPT (0.32) DHODHMAPTSMN1; SMN2TP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed