SCHEMBL6965327

SCHEMBL6965327

CC(C)c1nc(COCc2ccccc2)n(C)c1Cc1cc(Cl)cc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
VCP P55072 1/20 0.37
TACR1 P25103 5/20 0.37
CCR2 P41597 2/20 0.36
CCR5 P51681 2/20 0.36
TDP1 Q9NUW8 1/20 0.35
DHODH Q02127 2/20 0.35
RHEB Q15382 1/20 0.34
TSHR P16473 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PTGER1 P34995 1/20 0.33
F2RL3 Q96RI0 1/20 0.33
LTB4R Q15722 1/20 0.33
PSD A5PKW4 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957059 0.92 CCR2 (0.41) VCPTACR1CCR2CCR5TDP1
SCHEMBL6969238 0.80 VCP (0.38) VCPTACR1TDP1DHODHRHEB
SCHEMBL6961156 0.79 RHEB (0.37) VCPTACR1TDP1DHODHRHEB
SCHEMBL6969892 0.78 CCR2 (0.39) CCR2CCR5RHEB
SCHEMBL8099901 0.78 CCR2 (0.41) CCR2CCR5
SCHEMBL6973294 0.77 CCR2 (0.38) CCR2CCR5
SCHEMBL27410677 0.77 TDP1 (0.34) VCPTACR1TDP1DHODHRHEB
SCHEMBL6966825 0.75 VCP (0.43) VCPRHEBTSHRNPC1RAB9A
SCHEMBL6962017 0.74 TDP1 (0.39) VCPTACR1CCR2CCR5TDP1
SCHEMBL6960290 0.74 CCR2 (0.43) CCR2CCR5TDP1RHEBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed