SCHEMBL6969892

SCHEMBL6969892

CC(C)c1nc(CO)n(C)c1Cc1cc(Cl)cc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.39
CCR5 P51681 1/20 0.39
RHEB Q15382 1/20 0.32
GCGR P47871 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960290 0.87 CCR2 (0.43) CCR2CCR5RHEB
SCHEMBL8099901 0.86 CCR2 (0.41) CCR2CCR5
SCHEMBL6973911 0.81 CCR2 (0.41) CCR2CCR5
SCHEMBL6973294 0.80 CCR2 (0.38) CCR2CCR5
SCHEMBL6965327 0.78 VCP (0.37) CCR2CCR5RHEB
SCHEMBL6163272 0.74 HSP90B1 (0.33) GCGR
SCHEMBL6973358 0.72 HTR6 (0.31) CCR2CCR5GCGR
SCHEMBL6957943 0.72 GCGR (0.30) GCGR
SCHEMBL6957059 0.70 CCR2 (0.41) CCR2CCR5
SCHEMBL7083876 0.67 HSD11B1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed