SCHEMBL6960290

SCHEMBL6960290

CC(C)c1nc(CO)n(C)c1Cc1cccc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.43
CCR5 P51681 1/20 0.43
PDE5A O76074 1/20 0.40
PDE9A O76083 1/20 0.40
PDE1A P54750 1/20 0.40
PDE1B Q01064 1/20 0.40
PDE1C Q14123 1/20 0.40
PNMT P11086 1/20 0.39
GABRP O00591 2/20 0.37
GABRD O14764 2/20 0.37
GABRA1 P14867 2/20 0.37
GABRB1 P18505 2/20 0.37
GABRG2 P18507 2/20 0.37
GABRB3 P28472 2/20 0.37
GABRA5 P31644 2/20 0.37
GABRA3 P34903 2/20 0.37
GABRA2 P47869 2/20 0.37
GABRB2 P47870 2/20 0.37
GABRA4 P48169 2/20 0.37
GABRE P78334 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969892 0.87 CCR2 (0.39) CCR2CCR5RHEB
SCHEMBL6957059 0.82 CCR2 (0.41) CCR2CCR5PDE5APDE9APDE1A
SCHEMBL6969476 0.74 MEN1 (0.39) MAPTTDP1
SCHEMBL6965327 0.74 VCP (0.37) CCR2CCR5TSHRRHEBTDP1
SCHEMBL8099901 0.74 CCR2 (0.41) CCR2CCR5
SCHEMBL6968903 0.71 MEN1 (0.43) TSHRMAPTTDP1
SCHEMBL5749533 0.69 CCR2 (0.47) CCR2CCR5PDE5APDE9APDE1A
SCHEMBL6973294 0.69 CCR2 (0.38) CCR2CCR5
SCHEMBL6973911 0.69 CCR2 (0.41) CCR2CCR5PDE5APDE9APDE1A
SCHEMBL6975192 0.68 TDP1 (0.43) CCR2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed