SCHEMBL6965768

SCHEMBL6965768

CC(C)(C)[Si](C)(C)OCc1nccn1COCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DUT P33316 1/20 0.38
TSHR P16473 1/20 0.34
ADORA2A P29274 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ATP4A P20648 1/20 0.32
ATP4B P51164 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
AGER Q15109 1/20 0.32
MAPT P10636 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
KDM4E B2RXH2 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
GABRA1 P14867 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23053628 0.88 LTA4H (0.35) DUTTSHRHSP90AA1MEN1KMT2A
SCHEMBL18839693 0.86 HSP90AA1 (0.46) HSP90AA1HSD17B10MEN1KMT2ACYP1A2
SCHEMBL6973480 0.77 TSHR (0.41) TSHRHSP90AA1ATP4AATP4BCYP1A2
SCHEMBL28528886 0.77 ADRA2B (0.37) DUTTSHRADORA2AMEN1KMT2A
SCHEMBL1315036 0.74 IDO1 (0.46) TSHRCYP2D6MAPTTDP1L3MBTL1
SCHEMBL10434937 0.74 TSHR (0.44) TSHRHSD17B10MEN1KMT2AATP4A
SCHEMBL20518683 0.74 FPR2 (0.40) DUT
SCHEMBL23053629 0.73 DUT (0.35) DUTMEN1KMT2A
SCHEMBL25712857 0.73 DGAT1 (0.33) DUT
SCHEMBL7408576 0.72 CYP2D6 (0.42) TSHRHSP90AA1KMT2ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed