SCHEMBL6966022

SCHEMBL6966022

CC(C)c1nc(COC(N)=O)n(Cc2ccccn2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.36
PLA2G2A P14555 1/20 0.34
SLC16A3 O15427 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
MAPT P10636 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
XIAP P98170 1/20 0.33
BIRC2 Q13490 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TP53 P04637 1/20 0.33
P2RX3 P56373 1/20 0.32
RHEB Q15382 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7081501 0.93 NPC1 (0.38) ADRA1DPLA2G2ASLC16A3NPC1RAB9A
SCHEMBL7081480 0.93 ADRA1D (0.34) ADRA1DPLA2G2ASLC16A3NPC1RAB9A
SCHEMBL7078972 0.92 SLC16A3 (0.35) ADRA1DSLC16A3NPC1RAB9AMAPT
SCHEMBL7084635 0.91 ADRA1D (0.35) ADRA1DPLA2G2ASLC16A3CTSSCTSK
SCHEMBL6972378 0.91 TP53 (0.35) NPC1RAB9AMAPTCTSSCTSK
SCHEMBL7082317 0.90 PLA2G2A (0.36) PLA2G2ANPC1RAB9ATLR7SMN1; SMN2
SCHEMBL6967024 0.90 ALDH1A1 (0.35) PLA2G2ANPC1RAB9AMAPTTLR7
SCHEMBL8100819 0.90 HSP90B1 (0.33) ADRA1DNPC1RAB9AMAPTCTSS
SCHEMBL6972647 0.90 ADRA1D (0.34) ADRA1DPLA2G2ASLC16A3TLR7SMN1; SMN2
SCHEMBL6965296 0.90 NPC1 (0.38) SLC16A3NPC1RAB9AMAPTCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed