SCHEMBL6965296

SCHEMBL6965296

CNC(=O)OCc1nc(C(C)C)c(Sc2cc(Cl)cc(Cl)c2)n1Cc1ccccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
ENPP2 Q13822 1/20 0.34
LMNA P02545 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PTGER1 P34995 1/20 0.34
TOP2A P11388 1/20 0.33
TOP2B Q02880 1/20 0.33
TP53 P04637 1/20 0.33
SLC16A3 O15427 1/20 0.33
P2RX3 P56373 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082819 0.93 NPC1 (0.43) NPC1RAB9AMAPTSMN1; SMN2ENPP2
SCHEMBL7078972 0.91 SLC16A3 (0.35) NPC1RAB9AMAPTSMN1; SMN2MEN1
SCHEMBL6965963 0.90 TOP2A (0.40) NPC1RAB9AMAPTSMN1; SMN2ENPP2
SCHEMBL7084180 0.90 S1PR3 (0.39) NPC1RAB9ASMN1; SMN2ENPP2LMNA
SCHEMBL7077736 0.90 ALDH1A1 (0.33) NPC1RAB9AMAPTSMN1; SMN2MEN1
SCHEMBL6966022 0.90 ADRA1D (0.36) NPC1RAB9AMAPTSMN1; SMN2MEN1
SCHEMBL7081110 0.87 S1PR3 (0.39) NPC1RAB9AMAPTSMN1; SMN2ENPP2
SCHEMBL6961504 0.86 ENPP2 (0.35) ENPP2LMNAMEN1KMT2ATOP2A
SCHEMBL7087678 0.85 MEN1 (0.33) NPC1RAB9AMAPTSMN1; SMN2MEN1
SCHEMBL7082873 0.85 CFTR (0.40) NPC1RAB9AMAPTSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed