SCHEMBL6974348

SCHEMBL6974348

CCn1c(CCCOCc2ccccc2)nc(C(C)C)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.34
TLR7 Q9NYK1 4/20 0.33
TDP1 Q9NUW8 2/20 0.33
HRH4 Q9H3N8 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
TLR8 Q9NR97 1/20 0.32
ADORA1 P30542 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
PKM P14618 1/20 0.31
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30
VCP P55072 1/20 0.30
TACR1 P25103 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960981 0.90 TLR8 (0.33) TLR7TDP1HRH4HRH3TLR8
SCHEMBL6966496 0.89 VCP (0.37) TDP1L3MBTL1VCPTACR1
SCHEMBL6972963 0.89 GSK3B (0.38) GSK3BTLR7TDP1HRH4HRH3
SCHEMBL6975492 0.89 HRH4 (0.35) GSK3BTDP1HRH4HRH3MEN1
SCHEMBL6972834 0.86 TLR8 (0.35) TLR7TDP1TLR8MEN1KMT2A
SCHEMBL6974526 0.84 TDP1 (0.32) TLR7TDP1TLR8VCP
SCHEMBL7084679 0.83 TDP1 (0.36) GSK3BTLR7TDP1
SCHEMBL6964734 0.82 TDP1 (0.33) TDP1HRH4HRH3VCPTACR1
SCHEMBL14439828 0.82 TDP1 (0.40) TDP1KMT2AL3MBTL1VCPTACR1
SCHEMBL6972304 0.82 HSP90B1 (0.37) TLR7TDP1MEN1KMT2AVCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed