SCHEMBL7079909

SCHEMBL7079909

CC(C)c1nc(CO)n(Cc2ccncc2)c1Sc1cccc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.36
TDP1 Q9NUW8 2/20 0.35
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KCNH2 Q12809 1/20 0.33
POLB P06746 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE4B Q07343 1/20 0.33
TP53 P04637 2/20 0.32
KDM4E B2RXH2 2/20 0.32
RXFP1 Q9HBX9 1/20 0.32
GRM5 P41594 1/20 0.32
HTR6 P50406 2/20 0.32
ROCK2 O75116 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959029 0.92 IDO1 (0.35) IDO1TDP1CSNK2A2CSNK2BALDH1A1
SCHEMBL6975192 0.92 TDP1 (0.43) TDP1ALDH1A1POLBMEN1KMT2A
SCHEMBL5852651 0.90 KCNH2 (0.35) IDO1TDP1KCNH2MEN1KMT2A
SCHEMBL7083480 0.90 TLR8 (0.37) IDO1TDP1CSNK2A2CSNK2BALDH1A1
SCHEMBL6970034 0.90 ALDH1A1 (0.40) TDP1ALDH1A1SMN1; SMN2KMT2ATP53
SCHEMBL5031006 0.90 SLC2A4 (0.33) MEN1KMT2APIM1PIM3
SCHEMBL6967360 0.90 IDO1 (0.36) IDO1TDP1CSNK2A2CSNK2BALDH1A1
SCHEMBL8109545 0.89 GRIN1 (0.36) ALDH1A1MEN1KMT2ATP53KDM4E
SCHEMBL7084720 0.88 HTR3E (0.40) IDO1TDP1CSNK2A2CSNK2BALDH1A1
SCHEMBL7078348 0.88 SMN1; SMN2 (0.36) TDP1ALDH1A1SMN1; SMN2POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed