SCHEMBL6967975

SCHEMBL6967975

N=C(Nc1ccc(CCCNCc2cccc(Cl)c2)cc1)c1cccs1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 5/20 0.57
NOS1 P29475 4/20 0.57
NOS2 P35228 4/20 0.57
CHRM2 P08172 1/20 0.48
HTT P42858 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SLC2A1 P11166 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
KMT2A Q03164 1/20 0.42
CNR1 P21554 1/20 0.41
MARS1 P56192 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29558856 0.94 NOS3 (0.64) NOS3NOS1NOS2CHRM2HTT
SCHEMBL122445 0.94 NOS3 (0.64) NOS3NOS1NOS2CHRM2HTT
Hydrochloric Acid SCHEMBL31114391 0.93 NOS3 (0.65) NOS3NOS1NOS2CHRM2HTT
SCHEMBL6962188 0.86 SIGMAR1 (0.54) CHRM2SMN1; SMN2NPC1RAB9ASLC2A1
SCHEMBL6967589 0.85 NOS3 (0.59) NOS3NOS1NOS2CHRM2HTT
SCHEMBL18994883 0.85 NOS3 (0.42) NOS3NOS1NOS2HTTSMN1; SMN2
SCHEMBL15499648 0.84 NOS3 (0.51) NOS3NOS1NOS2HTTSMN1; SMN2
SCHEMBL6962276 0.82 NPC1 (0.52) NOS3NOS1NOS2HTTSMN1; SMN2
SCHEMBL6962883 0.82 NOS3 (0.49) NOS3NOS1NOS2SMN1; SMN2NPC1
SCHEMBL6961265 0.81 NOS1 (0.48) NOS3NOS1NOS2SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES Astra Aktiebolag (SE) 1996-05-29 EP claimed
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed