SCHEMBL7079263

SCHEMBL7079263

CC(C)c1nc(CN(C)C)n(Cc2ccccn2)c1Sc1cccc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
POLB P06746 1/20 0.39
GRM5 P41594 1/20 0.36
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
KDM4E B2RXH2 3/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
PKM P14618 1/20 0.35
ALDH1A1 P00352 4/20 0.35
KMT2A Q03164 3/20 0.35
MAPT P10636 2/20 0.35
PPP1CA P62136 1/20 0.35
TDP1 Q9NUW8 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969004 0.92 CYP1A2 (0.33) SLC6A2SLC6A4SLC6A3GRIN1GRIN2B
SCHEMBL7083143 0.89 GABRA1 (0.34) GRIN1GRIN2BALDH1A1CYP1A2CYP2D6
SCHEMBL6966820 0.89 GRIN1 (0.38) GRIN1GRIN2BKDM4EKMT2ASLC6A9
SCHEMBL7079929 0.89 GRM5 (0.38) POLBGRM5GRIN1GRIN2BKDM4E
SCHEMBL6962202 0.89 GRM5 (0.38) SLC6A2SLC6A4SLC6A3GRM5GRIN1
SCHEMBL6961462 0.87 GRIN1 (0.37) POLBGRM5GRIN1GRIN2BKDM4E
SCHEMBL6967528 0.87 GRM5 (0.36) GRM5GRIN1GRIN2BKDM4EL3MBTL1
SCHEMBL7082472 0.87 ALDH1A1 (0.37) GRM5GRIN1GRIN2BKDM4EL3MBTL1
SCHEMBL6969433 0.86 KMT2A (0.38) GRM5GRIN1GRIN2BKDM4EL3MBTL1
SCHEMBL6963923 0.85 POLB (0.44) SLC6A2SLC6A4SLC6A3POLBGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed