SCHEMBL6969304

SCHEMBL6969304

CCn1c(CCOC(C)=O)nc(C(C)C)c1Sc1cccc(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX12 P18054 1/20 0.36
SLC6A9 P48067 4/20 0.36
TP53 P04637 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
AKR1B1 P15121 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
TLR8 Q9NR97 1/20 0.34
NTRK1 P04629 1/20 0.34
NTRK2 Q16620 1/20 0.34
HPGD P15428 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7086454 0.92 ALOX12 (0.35) ALOX12SLC6A9TP53RXFP1AKR1B1
SCHEMBL6975636 0.91 ALOX12 (0.36) ALOX12SLC6A9TP53RXFP1AKR1B1
SCHEMBL7081639 0.90 ALOX12 (0.38) ALOX12SLC6A9TP53RXFP1AKR1B1
SCHEMBL6968155 0.90 TLR8 (0.34) TLR8KDM4E
SCHEMBL6974529 0.89 DHODH (0.34) SLC6A9MEN1ALDH1A1MAPTKMT2A
SCHEMBL6960486 0.88 IDO1 (0.34) ALOX12SLC6A9TP53RXFP1AKR1B1
SCHEMBL8116257 0.88 MEN1 (0.39) TP53MEN1ALDH1A1MAPTKMT2A
SCHEMBL6974700 0.86 ALOX12 (0.35) ALOX12SLC6A9TP53RXFP1AKR1B1
SCHEMBL6964051 0.85 IRAK4 (0.35) MEN1MAPTKMT2A
SCHEMBL7086211 0.85 ALDH1A1 (0.39) TP53MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed