SCHEMBL7086211

SCHEMBL7086211

CC(=O)OCCc1nc(C(C)C)c(Sc2cccc(Cl)c2)n1Cc1cccnc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
MCL1 Q07820 4/20 0.37
TP53 P04637 1/20 0.35
NPC1 O15118 2/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
GABRA5 P31644 3/20 0.33
GABRA1 P14867 2/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084645 0.93 ALDH1A1 (0.38) ALDH1A1LMNAMCL1TP53NPC1
SCHEMBL6973316 0.93 ALDH1A1 (0.39) ALDH1A1LMNAMCL1TP53NPC1
SCHEMBL6967425 0.92 ALDH1A1 (0.40) ALDH1A1LMNATP53NPC1GRIN1
SCHEMBL6960486 0.92 IDO1 (0.34) LMNATP53KMT2A
SCHEMBL7084562 0.90 KDM4E (0.37) ALDH1A1GABRA5GABRA1MEN1KMT2A
SCHEMBL6973497 0.88 ALDH1A1 (0.38) ALDH1A1LMNAMCL1TP53GRIN1
SCHEMBL8345861 0.87 LMNA (0.42) ALDH1A1LMNATP53GRIN1GRIN2B
SCHEMBL7085996 0.87 ALDH1A1 (0.39) ALDH1A1LMNATP53NPC1GRIN1
SCHEMBL6968344 0.87 ALDH1A1 (0.41) ALDH1A1LMNATP53NPC1GRIN1
SCHEMBL6972580 0.87 GRIN1 (0.36) GRIN1GRIN2BMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed