SCHEMBL6969489

SCHEMBL6969489

CC(C)c1nc(CN=C(N)N)n(Cc2cccnc2)c1Sc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
HPGD P15428 2/20 0.37
TLR7 Q9NYK1 5/20 0.36
MAPK1 P28482 2/20 0.36
POLB P06746 1/20 0.36
ALOX5AP P20292 1/20 0.35
SRC P12931 1/20 0.34
KDM4E B2RXH2 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
RECQL P46063 1/20 0.32
BLM P54132 1/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6962312 0.89 HTR3E (0.40) ALDH1A1HPGDSRCKDM4E
SCHEMBL6963828 0.89 GRIN1 (0.37) TLR7SRC
SCHEMBL6967507 0.89 PIM1 (0.34) ALDH1A1TLR7ALOX5APKDM4EGSK3B
SCHEMBL7078779 0.89 ADRA1D (0.35) ALDH1A1HPGDTLR7MAPK1POLB
SCHEMBL7081093 0.89 GRIN1 (0.37) HPGDTLR7ALOX5APSRC
SCHEMBL6972848 0.88 TLR7 (0.38) ALDH1A1TLR7MAPK1ALOX5APSRC
SCHEMBL7081083 0.88 ALOX5AP (0.37) ALDH1A1TLR7MAPK1POLBALOX5AP
SCHEMBL7081149 0.86 TLR7 (0.39) ALDH1A1TLR7MAPK1ALOX5APSRC
SCHEMBL7087890 0.86 TLR7 (0.41) ALDH1A1TLR7MAPK1ALOX5APSRC
SCHEMBL8109122 0.85 RECQL (0.47) ALDH1A1HPGDRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed